SCHEMBL21115031

SCHEMBL21115031

C=N[C@@H](Cc1ccccc1)c1nnc(-c2ccccc2)o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
GAA P10253 3/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TACR1 P25103 1/20 0.48
HPGD P15428 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
TSHR P16473 2/20 0.46
GPR55 Q9Y2T6 1/20 0.46
LMNA P02545 3/20 0.45
HTT P42858 2/20 0.45
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
HDAC6 Q9UBN7 2/20 0.43
EGFR P00533 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13828053 0.77 GAA (0.54) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL15047148 0.77 GAA (0.54) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL12527472 0.77 ALDH1A1 (0.56) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL12525246 0.77 ALDH1A1 (0.56) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL20204206 0.70 TACR1 (0.74) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL18167908 0.70 TACR1 (0.74) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL14858632 0.70 TACR1 (0.56) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL14762858 0.70 TACR1 (0.56) ALDH1A1GAAL3MBTL1TACR1HPGD
SCHEMBL14762860 0.70 TACR1 (0.56) ALDH1A1GAAL3MBTL1TACR1HPGD
Trifluoroacetic Acid SCHEMBL14763161 0.69 TACR1 (0.52) ALDH1A1GAAL3MBTL1TACR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3501546-A2 CYSTEINE DRUG CONJUGATES AND USE OF SAME Seattle Genetics, Inc. (US) 2019-06-26 EP disclosed