SCHEMBL21115562

SCHEMBL21115562

OB(O)c1ccc2c3c(cccc13)C1(c3ccccc3-c3ccccc31)c1ncccc1-2

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19974226 0.85 ESR1 (0.34) PDK2KMT2AESR1ESR2
SCHEMBL21110617 0.85 PDK2 (0.40) PDK2CYP1A2CYP2C19KMT2A
SCHEMBL19980421 0.81 CYP1A2 (0.41) CYP1A2KMT2A
SCHEMBL21113542 0.80 CYP11B1 (0.32) PDK2
SCHEMBL19980423 0.77 ALDH1A1 (0.39) PDK2CYP1A2CYP2C19KMT2AESR1
SCHEMBL19567023 0.77 ALDH1A1 (0.39) PDK2CYP1A2CYP2C19KMT2AESR1
SCHEMBL30322773 0.76 KMT2A (0.41) PDK2CYP1A2CYP2C19KMT2AESR1
SCHEMBL19009208 0.76 KMT2A (0.41) PDK2CYP1A2CYP2C19KMT2AESR1
SCHEMBL29739834 0.76 CRHBP (0.36) PDK2
SCHEMBL28767222 0.76 CRHBP (0.36) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11447464-B2 Compounds with spirobifluorene-structures MERCK PATENT GMBH (DE) 2022-09-20 US disclosed
US-20190194164-A1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES MERCK PATENT GMBH (DE) 2019-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11447464-B2 Compounds with spirobifluorene-structures SLCO1B3, SLCO4C1, SLCO1B1 PDK2 835/4885CYP1A2 787/4885CYP2C19 844/4885
US-20190194164-A1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES SLCO1B3, SLCO4C1, SLCO1B1 PDK2 835/4885CYP1A2 787/4885CYP2C19 844/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.