SCHEMBL211156

SCHEMBL211156

COC(=O)CC[C@@H](COC(=O)Nc1cc2ccccc2cn1)N(NCc1cccc(F)c1F)C(C)=O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.34
NOTUM Q6P988 1/20 0.33
ABL1 P00519 4/20 0.32
MAPK1 P28482 3/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
PIN1 Q13526 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAP4K1 Q92918 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
NTRK1 P04629 1/20 0.30
KMT2A Q03164 1/20 0.30
LMNA P02545 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30
MET P08581 1/20 0.30
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211133 0.95 CTSK (0.35) CTSKNOTUMABL1MAPK1PKM
SCHEMBL211083 0.95 CTSK (0.35) CTSKNOTUMABL1MAPK1PKM
SCHEMBL212049 0.93 ABL1 (0.33) ABL1MAPK1MET
SCHEMBL212477 0.93 CTSK (0.35) CTSKNOTUMABL1PIN1ALDH1A1
SCHEMBL209966 0.92 CTSK (0.34) CTSKNOTUMABL1MAPK1PKM
SCHEMBL4348546 0.91 CTSK (0.36) CTSKNOTUMABL1MAPK1PKM
SCHEMBL4347816 0.91 CTSK (0.36) CTSKNOTUMABL1MAPK1PKM
SCHEMBL214678 0.90 CTSK (0.36) CTSKNOTUMABL1PIN1ALDH1A1
SCHEMBL212192 0.90 CTSK (0.36) CTSKNOTUMABL1PIN1ALDH1A1
SCHEMBL215415 0.89 CTSK (0.36) CTSKNOTUMABL1PIN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US claimed
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed