SCHEMBL21132204

SCHEMBL21132204

Cc1ccc2c(c1)CC(C(=O)Nc1ccccn1)Cc1nnc(C3CCCCC3)n1-2

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 20/20 0.53
AVPR2 P30518 4/20 0.53
KCNH2 Q12809 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20020537 0.76 NPY5R (0.53)
SCHEMBL22010639 0.76 NPY5R (0.53)
SCHEMBL5139794 0.69 RAB9A (0.65)
Hydrochloric Acid SCHEMBL27440821 0.68 RAB9A (0.64)
SCHEMBL27488421 0.68 RAB9A (0.63)
SCHEMBL29500941 0.68 AVPR1A (0.73) AVPR1AAVPR2KCNH2
SCHEMBL29500702 0.68 AVPR1A (1.00) AVPR1AAVPR2KCNH2
SCHEMBL28449068 0.67 AVPR1A (0.80) AVPR1AAVPR2KCNH2
SCHEMBL28449067 0.67 AVPR1A (0.80) AVPR1AAVPR2KCNH2
SCHEMBL29500594 0.67 AVPR1A (0.80) AVPR1AAVPR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019116325-A1 TRICYCLIC COMPOUNDS AS VASOPRESSIN V1A RECEPTOR ANTAGONISTS RICHTER GEDEON NYRT. (HU) 2019-06-20 WO disclosed