Bromide

Bromide

SCHEMBL2113280

Br.CCOC(=O)c1csc(-c2cccnc2)n1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 1/20 0.62
HDAC6 Q9UBN7 1/20 0.60
RAB9A P51151 4/20 0.57
GAA P10253 1/20 0.57
IRAK4 Q9NWZ3 7/20 0.57
CDC7 O00311 2/20 0.57
DBF4 Q9UBU7 2/20 0.57
CYP2E1 P05181 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2A6 P11509 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2B6 P20813 1/20 0.55
MAOA P21397 1/20 0.54
MAOB P27338 1/20 0.54
NPC1 O15118 3/20 0.54
MAPT P10636 2/20 0.54
POLB P06746 1/20 0.54
PKM P14618 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
RXFP1 Q9HBX9 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290229 0.99 HDAC2 (0.63) HDAC2HDAC6RAB9AGAAIRAK4
SCHEMBL12571448 0.84 HDAC6 (0.69) HDAC2HDAC6RAB9AGAAIRAK4
SCHEMBL2080499 0.84 RAB9A (0.68) RAB9AGAACDC7DBF4MAOA
SCHEMBL2080725 0.84 RAB9A (0.68) HDAC6RAB9AGAACDC7DBF4
SCHEMBL3435162 0.83 RAB9A (0.60) HDAC2RAB9AGAACDC7DBF4
SCHEMBL3435697 0.83 RAB9A (0.60) HDAC2RAB9AGAACDC7DBF4
Bromide SCHEMBL7221661 0.82 CYP19A1 (0.60) RAB9AGAANPC1MAPTNPSR1
SCHEMBL27538606 0.81 CYP19A1 (0.61) RAB9AGAANPC1MAPTNPSR1
Bromide SCHEMBL368927 0.81 CYP2E1 (0.52) HDAC2HDAC6RAB9AGAAIRAK4
SCHEMBL9126190 0.81 KMT2A (0.52) HDAC2HDAC6RAB9ACDC7DBF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides DDT, PTMS, ACHE HDAC2 305/4885HDAC6 692/4885RAB9A 717/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.