SCHEMBL21133715

SCHEMBL21133715

COc1cc(-c2ccnn2C)ccc1NI

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.54
BRD4 O60885 1/20 0.50
BRD3 Q15059 1/20 0.50
TTK P33981 2/20 0.46
GRM7 Q14831 1/20 0.42
P2RX7 Q99572 5/20 0.41
ICMT O60725 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PI4KA P42356 1/20 0.40
PIK3CG P48736 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17049306 0.82 BRD4 (0.50) LRRK2BRD4BRD3TTKGRM7
SCHEMBL28058890 0.82 GRM7 (0.56) LRRK2BRD4BRD3GRM7ICMT
SCHEMBL26545148 0.81 BRD4 (0.47) LRRK2BRD4BRD3TTKGRM7
SCHEMBL24497540 0.79 KDM5A (0.52) LRRK2BRD4BRD3TTKGRM7
SCHEMBL15652106 0.79 ALDH1A1 (0.59) LRRK2BRD4BRD3TTKGRM7
SCHEMBL31051265 0.78 BRD4 (0.47) LRRK2BRD4BRD3TTKGRM7
SCHEMBL27398722 0.78 BRD4 (0.47) LRRK2BRD4BRD3TTKGRM7
SCHEMBL16911970 0.76 BRD4 (0.51) LRRK2BRD4BRD3TTKGRM7
SCHEMBL26544695 0.75 BRD4 (0.46) LRRK2BRD4BRD3TTKGRM7
SCHEMBL28234703 0.75 KDM4E (0.47) BRD4BRD3GRM7ICMTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3110816-B1 N2-PHENYL-PYRIDO[3,4-D]PYRIMIDINE-2,8-DIAMINE DERIVATIVES AND THEIR USE AS MPS1 INHIBITORS CANCER RESEARCH TECH LTD (GB) 2019-06-19 EP disclosed