SCHEMBL21135205

SCHEMBL21135205

C=NNc1cc2nc(C(=O)NC3CCOCC3)cn2c(N2CCOCC2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.53
PIK3CA P42336 2/20 0.42
MTOR P42345 2/20 0.42
CNR2 P34972 3/20 0.38
NAPEPLD Q6IQ20 1/20 0.37
DPP4 P27487 1/20 0.37
DPP8 Q6V1X1 1/20 0.37
DPP9 Q86TI2 1/20 0.37
BRD4 O60885 2/20 0.34
SMYD3 Q9H7B4 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
GRIA1 P42261 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
DNM1L O00429 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21135203 0.85 ATR (0.45) ATRPIK3CAMTORCNR2NAPEPLD
SCHEMBL21055102 0.81 KDM4E (0.51) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL21055507 0.78 ATR (0.52) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL30312386 0.78 ATR (0.52) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL30312517 0.77 KDM4E (0.49) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL21055026 0.77 KDM4E (0.49) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL21055011 0.77 LMNA (0.51) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL30312410 0.77 LMNA (0.51) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL21135504 0.77 LMNA (0.51) ATRALDH1A1LMNAKDM4EMAPT
SCHEMBL30312523 0.77 LMNA (0.51) ATRALDH1A1LMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019113523-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF BAJJI ASHOK (US) 2019-06-13 WO disclosed