SCHEMBL21159124

SCHEMBL21159124

FC(F)(F)C1CCCCC(c2nnc3c(Cl)nccn23)C1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 11/20 0.37
NR1I2 O75469 1/20 0.37
ADORA3 P0DMS8 3/20 0.33
YTHDC1 Q96MU7 1/20 0.32
CCNE1 P24864 3/20 0.32
CDK2 P24941 3/20 0.32
CCNT1 O60563 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNA2 P20248 1/20 0.32
CCND1 P24385 1/20 0.32
CDK9 P50750 1/20 0.32
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21138374 0.99 HSD11B1 (0.35) HSD11B1NR1I2ADORA3YTHDC1IDO1
SCHEMBL21057270 0.85 ADORA3 (0.44) ADORA3
SCHEMBL21057273 0.85 ADORA3 (0.44) ADORA3
SCHEMBL21138331 0.84 HSD11B1 (0.47) HSD11B1NR1I2ADORA3CCNE1CDK2
SCHEMBL21138816 0.83 HSD11B1 (0.49) HSD11B1NR1I2ADORA3CCNE1CDK2
SCHEMBL21138249 0.83 HSD11B1 (0.45) HSD11B1NR1I2ADORA3CCNE1CDK2
SCHEMBL21138894 0.81 HSD11B1 (0.34) HSD11B1
SCHEMBL19917049 0.80 HSD11B1 (0.37) HSD11B1NR1I2ADORA3CCNE1CDK2
SCHEMBL21057446 0.80 HSD11B1 (0.37) HSD11B1NR1I2ADORA3CCNE1CDK2
SCHEMBL30396230 0.80 HSD11B1 (0.37) HSD11B1NR1I2ADORA3CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3505171-A1 BICYCLIC NITROGENATED HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2019-07-03 EP disclosed