SCHEMBL21159366

SCHEMBL21159366

CC1CCCC(N(N)c2ncnc(N)c2N)C1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 10/20 0.49
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
JAK1 P23458 6/20 0.36
CYP3A4 P08684 1/20 0.36
JAK2 O60674 2/20 0.35
HTT P42858 1/20 0.33
LIMK1 P53667 2/20 0.33
MAP4K4 O95819 1/20 0.32
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
TYK2 P29597 1/20 0.30
MCHR1 Q99705 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21159571 0.83 JAK3 (0.46) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL21159272 0.83 JAK3 (0.42) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL19916990 0.83 JAK3 (0.42) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL21159280 0.82 JAK1 (0.37) JAK3MEN1KMT2AJAK1JAK2
SCHEMBL21159262 0.82 MAP4K4 (0.36) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL21159292 0.79 JAK3 (0.33) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL21159109 0.79 PAK1 (0.35) JAK3JAK1
SCHEMBL21159572 0.79 MAP4K4 (0.36) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL21159353 0.79 JAK3 (0.34) JAK3MEN1KMT2AJAK1CYP3A4
SCHEMBL19917011 0.79 MAP4K4 (0.36) JAK3MEN1KMT2AJAK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3505171-A1 BICYCLIC NITROGENATED HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2019-07-03 EP disclosed