SCHEMBL21164006

SCHEMBL21164006

Nc1ccc(-c2ccnc(N)n2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.70
AURKA O14965 2/20 0.70
PRKACA P17612 1/20 0.70
ADORA2A P29274 1/20 0.70
RAB9A P51151 4/20 0.61
NPC1 O15118 2/20 0.61
KMO O15229 1/20 0.59
KDM4E B2RXH2 5/20 0.59
ALDH1A1 P00352 5/20 0.59
MAPT P10636 3/20 0.59
HSP90AB1 P08238 1/20 0.56
PTK2 Q05397 1/20 0.56
CDK2 P24941 2/20 0.51
CHUK O15111 1/20 0.51
PDPK1 O15530 1/20 0.51
RPS6KB1 P23443 1/20 0.51
KDR P35968 1/20 0.51
TGFBR1 P36897 1/20 0.51
SYK P43405 1/20 0.51
JAK3 P52333 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12821368 0.83 HSP90AA1 (0.66) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL474287 0.83 HSP90AA1 (0.66) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL2994671 0.83 HSP90AA1 (0.66) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL3412705 0.83 KMO (0.66) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL17200126 0.83 HSP90AA1 (0.66) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL8313279 0.83 HSP90AA1 (0.66) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL12176972 0.83 HSP90AA1 (0.92) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL3454021 0.83 KMO (0.60) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL15876512 0.83 MEN1 (0.55) HSP90AA1AURKAPRKACAADORA2ARAB9A
SCHEMBL2684649 0.83 HSP90AA1 (0.70) HSP90AA1AURKAPRKACAADORA2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111065635-A Novel pyrimidine derivatives as MTH1 inhibitors 无锡安万生物科技有限公司 2020-04-24 CN claimed
CN-111065635-B Novel pyrimidine derivatives as MTH1 inhibitors 无锡安万生物科技有限公司 2022-07-22 CN disclosed
CN-111065635-A Novel pyrimidine derivatives as MTH1 inhibitors 无锡安万生物科技有限公司 2020-04-24 CN disclosed
WO-2019134082-A1 NOVEL PYRIMIDINE DERIVATIVES AS MTH1 INHIBITORS WUXI ADVANT BIOTECHNOLOGY CO., LTD. (CN) 2019-07-11 WO disclosed