SCHEMBL21165038

SCHEMBL21165038

Cc1ccc(Cc2ccc(-c3ccncc3)nc2)cn1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 16/20 0.64
CYP11B2 P19099 16/20 0.64
CYP3A4 P08684 2/20 0.52
MAPK1 P28482 1/20 0.41
GRM5 P41594 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18459203 0.84 CYP11B1 (0.54) CYP11B1CYP11B2CYP3A4
SCHEMBL12533585 0.79 RAB9A (0.58) CYP11B1CYP11B2CYP3A4MAPK1
SCHEMBL2718952 0.78 CYP11B1 (1.00) CYP11B1CYP11B2CYP3A4
SCHEMBL13658677 0.77 CYP11B1 (0.59) CYP11B1CYP11B2CYP3A4
SCHEMBL18525554 0.77 CYP11B1 (0.47) CYP11B1CYP11B2CYP3A4
SCHEMBL13658668 0.76 CYP11B1 (0.58) CYP11B1CYP11B2CYP3A4
SCHEMBL14355101 0.75 CYP11B1 (0.54) CYP11B1CYP11B2CYP3A4MAPK1
SCHEMBL14355099 0.75 CYP11B1 (0.57) CYP11B1CYP11B2CYP3A4CYP2A6
SCHEMBL12880434 0.75 MAPK1 (0.48) CYP3A4MAPK1GRM5CYP2A6
SCHEMBL18459206 0.75 CYP11B1 (0.60) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023275357-A1 CASPASE-2 INHIBITOR COMPOUNDS Kintsugi Therapeutics S.L. (ES) 2023-01-05 WO disclosed
EP-4112631-A1 CASPASE-2 INHIBITOR COMPOUNDS Kintsugi Therapeutics S.L. (ES) 2023-01-04 EP disclosed
US-10355284-B2 Composition, method of preparing the composition, electrode including the composition, and fuel cell including the electrode SAMSUNG ELECTRONICS CO., LTD. (KR) 2019-07-16 US disclosed