SCHEMBL21167480

SCHEMBL21167480

CCCn1cc(-c2cnc(N)c(NCc3ccc4nccn4c3)n2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 7/20 0.47
CSF1R P07333 1/20 0.46
MAPK1 P28482 1/20 0.39
NAMPT P43490 1/20 0.39
KEAP1 Q14145 1/20 0.38
LDHA P00338 1/20 0.37
LDHB P07195 1/20 0.37
TYRO3 Q06418 1/20 0.36
PAK1 Q13153 1/20 0.36
NQO2 P16083 1/20 0.36
ATR Q13535 1/20 0.35
SYK P43405 1/20 0.35
PIK3CD O00329 1/20 0.34
PIP5K1C O60331 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PI4KA P42356 1/20 0.34
PIK3CG P48736 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22475658 0.93 CSF1R (0.46) METCSF1RMAPK1KEAP1LDHA
SCHEMBL21167404 0.91 MET (0.58) METCSF1RKEAP1LDHALDHB
SCHEMBL24590985 0.90 MET (0.46) METCSF1RTYRO3SYKPIK3CD
SCHEMBL22475990 0.90 MET (0.47) METCSF1RMAPK1NAMPTKEAP1
SCHEMBL21167421 0.89 CSF1R (0.59) METCSF1RMAPK1KEAP1LDHA
SCHEMBL24590986 0.86 MET (0.59) METCSF1RNAMPTKEAP1LDHA
SCHEMBL22475927 0.86 MET (0.43) METCSF1RKEAP1LDHALDHB
SCHEMBL23128064 0.85 MET (0.44) METCSF1RMAPK1NAMPTKEAP1
SCHEMBL21167673 0.84 CSF1R (0.45) METCSF1RMAPK1NAMPTKEAP1
SCHEMBL21167380 0.82 DYRK1A (0.44) METCSF1RNAMPTKEAP1LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3511330-A1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS Hutchison Medipharma Limited (CN) 2019-07-17 EP disclosed