SCHEMBL21170044

SCHEMBL21170044

Cc1cc(NCC(C)c2ccc(F)cc2)nnc1-c1cccc(C(N)=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.40
DHODH Q02127 1/20 0.39
MAPK14 Q16539 2/20 0.38
PARP1 P09874 3/20 0.38
MAP3K5 Q99683 1/20 0.38
FYN P06241 1/20 0.38
MAP2K4 P45985 1/20 0.37
CLK1 P49759 1/20 0.36
KDR P35968 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
LDHB P07195 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
ADAMTS4 O75173 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12287289 0.85 DPP4 (0.42) DPP4MAPK14PARP1FYNCLK1
SCHEMBL12287723 0.85 DPP4 (0.42) DPP4MAPK14PARP1FYNCLK1
SCHEMBL21170038 0.85 DPP4 (0.42) DPP4MAPK14PARP1FYNCLK1
SCHEMBL21170168 0.81 DPP4 (0.41) DPP4MAPK14PARP1FYNCLK1
SCHEMBL2558433 0.80 KDR (0.44) DHODHMAPK14PARP1MAP2K4CLK1
SCHEMBL21170045 0.80 PTGDR2 (0.43) MAPK14KDRPTGDR2PSEN1PSEN2
SCHEMBL12295523 0.80 DPP4 (0.48) DPP4PARP1FYNCLK1LDHB
SCHEMBL12295515 0.80 DPP4 (0.48) DPP4PARP1FYNCLK1LDHB
SCHEMBL19422102 0.78 FYN (0.40) DHODHPARP1MAP3K5FYNMAP2K4
SCHEMBL19422104 0.78 FYN (0.40) DHODHPARP1MAP3K5FYNMAP2K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed