SCHEMBL21170045

SCHEMBL21170045

Cc1cc(NCC(C)c2ccc(F)cc2)nnc1-c1cccc(C#N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.43
GABRG2 P18507 5/20 0.41
GABRB3 P28472 5/20 0.41
GABRA5 P31644 5/20 0.41
GABRA3 P34903 5/20 0.41
MAPK14 Q16539 2/20 0.39
KCNK3 O14649 1/20 0.39
MCHR1 Q99705 1/20 0.38
TRPA1 O75762 1/20 0.38
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
NPY5R Q15761 1/20 0.37
MAPK1 P28482 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21170143 0.83 GABRG2 (0.43) PTGDR2GABRG2GABRB3GABRA5GABRA3
SCHEMBL21170044 0.80 DPP4 (0.40) PTGDR2MAPK14PSEN1PSEN2APH1B
SCHEMBL12287314 0.80 TRPA1 (0.42) PTGDR2GABRG2GABRB3GABRA5GABRA3
SCHEMBL21170333 0.80 GABRG2 (0.44) PTGDR2GABRG2GABRB3GABRA5GABRA3
SCHEMBL21170118 0.72 NPY5R (0.40) NPY5R
SCHEMBL12287988 0.69 KCNH2 (0.44) GABRG2GABRB3GABRA5GABRA3ADORA2A
SCHEMBL11625379 0.67 CLK4 (0.45) GABRG2GABRB3GABRA5GABRA3TRPA1
SCHEMBL11634822 0.67 ADORA2A (0.41) PTGDR2GABRG2GABRB3GABRA5GABRA3
SCHEMBL11628595 0.67 ADORA2A (0.44) GABRG2GABRB3GABRA5GABRA3ADORA2A
SCHEMBL14734692 0.66 GABRG2 (0.36) GABRG2GABRB3GABRA5GABRA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed