SCHEMBL21170038

SCHEMBL21170038

CC(CNc1ccc(-c2cccc(C(N)=O)c2)nn1)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.42
HPGDS O60760 1/20 0.40
FYN P06241 1/20 0.39
LDHB P07195 1/20 0.39
CLK1 P49759 1/20 0.38
PARP1 P09874 3/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
PIK3CA P42336 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
ADAMTS4 O75173 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12287723 1.00 DPP4 (0.42) DPP4HPGDSFYNLDHBCLK1
SCHEMBL12287289 1.00 DPP4 (0.42) DPP4HPGDSFYNLDHBCLK1
SCHEMBL21170446 0.91 HPGDS (0.44) DPP4HPGDSFYNLDHBPARP1
SCHEMBL19422102 0.91 FYN (0.40) FYNLDHBPARP1PIK3CAMAPK8
SCHEMBL19422104 0.91 FYN (0.40) FYNLDHBPARP1PIK3CAMAPK8
SCHEMBL12286690 0.90 LDHB (0.47) FYNLDHBPARP1PIK3CAMAPK8
SCHEMBL21170136 0.90 LDHB (0.43) FYNLDHBPARP1MEN1KMT2A
SCHEMBL21170185 0.89 TRPM8 (0.41) LDHBTRPM8MEN1NPC1ALDH1A1
SCHEMBL21170091 0.89 MAP4K4 (0.38) FYNTRPM8MEN1NPC1ALDH1A1
SCHEMBL21170314 0.88 NPC1 (0.41) DPP4CLK1MEN1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed