SCHEMBL21170417

SCHEMBL21170417

C=C(N)c1ccc(F)c(-c2ccc(NCC(C)(C)c3ncccc3Cl)nn2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL1B P01584 7/20 0.36
NLRP3 Q96P20 1/20 0.36
NPC1 O15118 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
KMT2A Q03164 1/20 0.32
RELA Q04206 1/20 0.32
CDC7 O00311 1/20 0.30
ROCK2 O75116 1/20 0.30
PIM1 P11309 1/20 0.30
PRKACA P17612 1/20 0.30
CDK2 P24941 1/20 0.30
GSK3B P49841 1/20 0.30
HIPK2 Q9H2X6 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2560960 0.91 IL1B (0.36) IL1BNLRP3NPC1ALDH1A1MAPT
SCHEMBL12287239 0.82 IL1B (0.35) IL1BNLRP3KMT2A
SCHEMBL21170329 0.81 IL1B (0.34) IL1BNLRP3NPC1ALDH1A1MAPT
SCHEMBL15008937 0.78 PTK2 (0.36)
SCHEMBL14990448 0.77 NPC1 (0.37) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL15008831 0.77 RORC (0.35) SMN1; SMN2
SCHEMBL2564397 0.76 PDE4A (0.38) IL1BNLRP3
SCHEMBL15009090 0.74 RORC (0.35) MAPTMEN1KMT2AROCK2
SCHEMBL21170223 0.73 IL1B (0.34) IL1BNLRP3
SCHEMBL17690354 0.73 KCNH2 (0.33) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed