SCHEMBL211720

SCHEMBL211720

CN(C(=O)NCc1cccc(F)c1F)[C@@H](CCCOP(=O)(O)O)COC(=O)Nc1cc2ccccc2cn1.[NaH]

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.38
CTSK P43235 1/20 0.35
NOTUM Q6P988 1/20 0.33
NTRK1 P04629 1/20 0.31
MET P08581 1/20 0.31
MAOB P27338 1/20 0.31
PKM P14618 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
WNT1 P04628 1/20 0.30
GSK3B P49841 1/20 0.30
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL210233 0.99 PIN1 (0.38) PIN1CTSKNOTUMNTRK1MET
SCHEMBL210234 0.99 PIN1 (0.38) PIN1CTSKNOTUMNTRK1MET
SCHEMBL210235 0.99 PIN1 (0.38) PIN1CTSKNOTUMNTRK1MET
SCHEMBL210409 0.97 PIN1 (0.38) PIN1CTSKNOTUMNTRK1MET
SCHEMBL210408 0.97 PIN1 (0.38) PIN1CTSKNOTUMNTRK1MET
SCHEMBL210410 0.97 PIN1 (0.38) PIN1CTSKNOTUMNTRK1MET
SCHEMBL209916 0.93 PIN1 (0.34) PIN1CTSKMETMAOBMAPK1
SCHEMBL211719 0.93 CTSK (0.35) PIN1CTSKNOTUMNTRK1MET
SCHEMBL212719 0.92 CTSK (0.35) PIN1CTSKNOTUMNTRK1MET
SCHEMBL212721 0.92 CTSK (0.35) PIN1CTSKNOTUMNTRK1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed