SCHEMBL2117237

SCHEMBL2117237

CCCCCOC(=O)c1cccc2ccccc12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.73
MAPK1 P28482 3/20 0.73
CYP3A4 P08684 2/20 0.73
TP53 P04637 1/20 0.73
ALDH1A1 P00352 7/20 0.71
LMNA P02545 2/20 0.71
TDP1 Q9NUW8 2/20 0.66
L3MBTL1 Q9Y468 2/20 0.66
KDM4E B2RXH2 4/20 0.62
HSD17B10 Q99714 2/20 0.62
POLB P06746 1/20 0.62
HRH3 Q9Y5N1 2/20 0.62
CNR1 P21554 3/20 0.61
CNR2 P34972 3/20 0.61
CYP2C9 P11712 1/20 0.61
CDC25B P30305 2/20 0.58
DRD3 P35462 1/20 0.55
KDM4A O75164 1/20 0.54
KDM4C Q9H3R0 1/20 0.54
CDC25A P30304 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5709967 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL8665013 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL30295637 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL9288049 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL20100237 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL27721668 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL4407176 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL27729056 0.98 ALDH1A1 (0.74) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL27477086 0.97 ALDH1A1 (0.72) TSHRMAPK1CYP3A4TP53ALDH1A1
SCHEMBL9681013 0.97 ALDH1A1 (0.72) TSHRMAPK1CYP3A4TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170159189-A1 METHOD FOR PRODUCING 1,5-DIAMINONAPHTHALENE AND 1-AMINO-5-NITRONAPHTHALENE BY DIRECT ELECTROCHEMICAL AMINATION OF NON-ACTIVATED OR DEACTIVATED AROMATIC SYSTEMS ON BORON-DOPED DIAMOND ANODES COVESTRO DEUTSCHLAND AG (DE) 2017-06-08 US claimed
CN-104558085-B Naphthoic acid Pentamethylene. many hydrogen phenanthrene ester B and extracting method thereof and medicinal usage 吉林农业大学 2016-08-17 CN claimed
CN-104558085-A Naphthoic acid cyclopentanoperhydrophenanthrene ester B and extraction method and pharmaceutical application thereof UNIV JILIN AGRICULTURAL 2015-04-29 CN claimed
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDTJYLLAND (DK) 2013-05-16 US claimed
US-20120095048-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDT JYLLAND (DK) 2012-04-19 US claimed
EP-2398760-A1 ALLOSTERIC BINDING COMPOUNDS Aarhus Universitet (DK) 2011-12-28 EP claimed
WO-2010094289-A1 ALLOSTERIC BINDING COMPOUNDS AARHUS UNIVERSITET (DK) 2010-08-26 WO claimed
US-20170159189-A1 METHOD FOR PRODUCING 1,5-DIAMINONAPHTHALENE AND 1-AMINO-5-NITRONAPHTHALENE BY DIRECT ELECTROCHEMICAL AMINATION OF NON-ACTIVATED OR DEACTIVATED AROMATIC SYSTEMS ON BORON-DOPED DIAMOND ANODES COVESTRO DEUTSCHLAND AG (DE) 2017-06-08 US disclosed
CN-104558085-B Naphthoic acid Pentamethylene. many hydrogen phenanthrene ester B and extracting method thereof and medicinal usage 吉林农业大学 2016-08-17 CN disclosed
CN-104558085-B Naphthoic acid Pentamethylene. many hydrogen phenanthrene ester B and extracting method thereof and medicinal usage 吉林农业大学 2016-08-17 CN disclosed
CN-104558085-B Naphthoic acid Pentamethylene. many hydrogen phenanthrene ester B and extracting method thereof and medicinal usage 吉林农业大学 2016-08-17 CN disclosed
CN-104558085-A Naphthoic acid cyclopentanoperhydrophenanthrene ester B and extraction method and pharmaceutical application thereof UNIV JILIN AGRICULTURAL 2015-04-29 CN disclosed
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDTJYLLAND (DK) 2013-05-16 US disclosed
WO-2010094289-A1 ALLOSTERIC BINDING COMPOUNDS AARHUS UNIVERSITET (DK) 2010-08-26 WO disclosed
EP-0432910-B1 Process for producing highly pure 2, 6 naphthalene dicarboxylic acid MITSUBISHI GAS CHEMICAL CO (JP) 1995-06-14 EP disclosed
US-5326848-A Thermotropic liquid crystal polyester KURARAY CO., LTD. (JP) 1994-07-05 US disclosed
US-5068410-A Hydrolysis of 2,6-dimethyl naphthalene dicarboxylate in an aqueous solution using an aromatic polycarboxylic acid or anhydride as a catalyst MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1991-11-26 US disclosed
EP-0432910-A2 Process for producing highly pure 2, 6 naphthalene dicarboxylic acid MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1991-06-19 EP disclosed
US-4931420-A COLOR CHANGING LABELS, CHIPS FOR STORED FOODS, MEDICINES, BLOOD; RUPTURABLE CAPSULES CONTAINING DYE AND DEVELOPER MITSUI TOATSU CHEMICALS, INC. (JP) 1990-06-05 US disclosed
EP-0244219-A2 Temperature history indicator and its manufacture MITSUI TOATSU CHEMICALS, Inc. (JP) 1987-11-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120095048-A1 ALLOSTERIC BINDING COMPOUNDS GRIN2C, GRM2, GRIN2B TSHR 534/4885MAPK1 1555/4885CYP3A4 796/4885
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS GRIN2C, GRM2, GRIN2B TSHR 534/4885MAPK1 1555/4885CYP3A4 796/4885
US-20170159189-A1 METHOD FOR PRODUCING 1,5-DIAMINONAPHTHALENE AND 1-AMINO-5-NITRONAPHTHALENE BY DIRECT ELECTROCHEMICAL AMINATION OF NON-ACTIVATED OR DEACTIVATED AROMATIC SYSTEMS ON BORON-DOPED DIAMOND ANODES DAO, APEX1, DDAH1 TSHR 3769/4885MAPK1 812/4885CYP3A4 212/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.