SCHEMBL21174663

SCHEMBL21174663

COc1cc2cc(-c3cccc(-c4nc5ccccc5[nH]4)c3)ccc2cc1-n1ccnc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.57
CYP11B1 P15538 1/20 0.57
CYP11B2 P19099 1/20 0.57
KDM4E B2RXH2 5/20 0.46
NPC1 O15118 5/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
ALDH1A1 P00352 4/20 0.46
RAB9A P51151 4/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 3/20 0.43
HPSE Q9Y251 4/20 0.42
BACE1 P56817 2/20 0.41
BACE2 Q9Y5Z0 2/20 0.41
COMT P21964 1/20 0.41
HPGD P15428 3/20 0.41
TP53 P04637 2/20 0.41
HSD17B10 Q99714 2/20 0.41
AMY1A P0DUB6 2/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16148286 0.84 NPC1 (0.60) KDM4ENPC1SMN1; SMN2ALDH1A1RAB9A
SCHEMBL16147474 0.79 ALDH1A1 (0.54) KDM4ENPC1SMN1; SMN2ALDH1A1RAB9A
SCHEMBL21174653 0.78 KDM4E (0.55) CYP19A1CYP11B1CYP11B2KDM4ENPC1
SCHEMBL16158580 0.77 CYP19A1 (0.56) CYP19A1CYP11B1CYP11B2SMN1; SMN2ALDH1A1
SCHEMBL16148101 0.76 NPC1 (0.51) KDM4ENPC1SMN1; SMN2ALDH1A1RAB9A
SCHEMBL16147181 0.76 NPC1 (0.70) CYP11B1CYP11B2KDM4ENPC1SMN1; SMN2
SCHEMBL16148300 0.76 NPC1 (0.48) KDM4ENPC1SMN1; SMN2ALDH1A1RAB9A
SCHEMBL21174655 0.76 MMP2 (0.58) KDM4ENPC1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL16147757 0.75 KDM4E (0.55) KDM4ENPC1SMN1; SMN2ALDH1A1RAB9A
SCHEMBL4508354 0.75 CYP11B1 (1.00) CYP19A1CYP11B1CYP11B2KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3514147-A1 STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY University of Maryland, Baltimore (US) 2019-07-24 EP disclosed