SCHEMBL211772

SCHEMBL211772

CN(C(=O)NCc1cccc(F)c1F)[C@H](COC(=O)Nc1cc2ccccc2cn1)C[C@H](O)COP(=O)(O)O.[NaH]

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.40
NOTUM Q6P988 1/20 0.33
DYRK1A Q13627 3/20 0.32
GSK3B P49841 2/20 0.32
WNT1 P04628 1/20 0.32
NTRK1 P04629 1/20 0.31
MET P08581 1/20 0.31
CTSK P43235 1/20 0.31
MAOB P27338 1/20 0.31
MAPK1 P28482 2/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
RPS6KA1 Q15418 1/20 0.30
GCK P35557 2/20 0.30
RARA P10276 1/20 0.30
RARB P10826 1/20 0.30
RARG P13631 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211922 1.00 PIN1 (0.40) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL2840927 0.99 PIN1 (0.40) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL213747 0.99 PIN1 (0.40) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL212113 0.99 PIN1 (0.40) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL209908 0.99 PIN1 (0.40) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL2840914 0.94 PIN1 (0.34) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL4348511 0.94 PIN1 (0.34) PIN1NOTUMDYRK1AGSK3BWNT1
SCHEMBL211785 0.94 PIN1 (0.36) PIN1DYRK1AGSK3BWNT1MET
SCHEMBL2724097 0.94 PIN1 (0.36) PIN1DYRK1AGSK3BWNT1MET
SCHEMBL212784 0.93 PIN1 (0.34) PIN1NOTUMDYRK1AGSK3BWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed