SCHEMBL21177347

SCHEMBL21177347

O=C(NCCCO)c1cc(Br)ccc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.68
CYP1A2 P05177 1/20 0.66
CDK1 P06493 1/20 0.55
ALDH1A1 P00352 4/20 0.53
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA3 P07451 1/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA5A P35218 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
CA13 Q8N1Q1 1/20 0.53
CA14 Q9ULX7 1/20 0.53
CA5B Q9Y2D0 1/20 0.53
KDM4E B2RXH2 1/20 0.53
THRB P10828 1/20 0.51
HTT P42858 1/20 0.51
KMT2A Q03164 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177405 0.95 HPGD (0.66) HPGDCYP1A2CDK1ALDH1A1CA12
SCHEMBL2566261 0.83 HPGD (0.69) HPGDCYP1A2ALDH1A1KDM4ETHRB
SCHEMBL7223858 0.80 HPGD (0.68) HPGDCYP1A2ALDH1A1KDM4ETHRB
SCHEMBL2562980 0.79 CYP1A2 (0.70) HPGDCYP1A2ALDH1A1KDM4ETHRB
SCHEMBL20694515 0.78 HPGD (0.62) HPGDCYP1A2ALDH1A1CA1CA2
SCHEMBL5111555 0.77 P2RX7 (0.66) HPGDCYP1A2KMT2AMEN1P2RX7
SCHEMBL21977975 0.77 HPGD (0.78) HPGDCYP1A2ALDH1A1CA12CA1
SCHEMBL9778626 0.77 ALDH1A1 (0.68) HPGDCYP1A2ALDH1A1KDM4EKMT2A
SCHEMBL2564944 0.77 HPGD (0.61) HPGDCYP1A2ALDH1A1KDM4EHTT
SCHEMBL21177406 0.77 CDK1 (0.49) HPGDCYP1A2CDK1ALDH1A1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3740489-A1 PI4KIIIBETA INHIBITORS GlaxoSmithKline Intellectual Property Development Limited (GB) 2020-11-25 EP disclosed
WO-2019141694-A1 PI4KIIIBETA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-07-25 WO disclosed