SCHEMBL21182252

SCHEMBL21182252

Cc1c(-c2cnc(Cl)cn2)nc2ccc(C(F)(F)F)cn12

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 8/20 0.46
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC2A1 P11166 1/20 0.38
CYP11B1 P15538 4/20 0.37
CYP11B2 P19099 4/20 0.37
MCHR1 Q99705 1/20 0.37
GABRD O14764 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRA4 P48169 1/20 0.36
CYP1A2 P05177 1/20 0.36
USP7 Q93009 1/20 0.36
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK2 Q92630 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21182258 0.85 TRPA1 (0.41) TRPA1ALDH1A1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL19992608 0.83 TRPA1 (0.40) TRPA1SMN1; SMN2CYP11B1CYP11B2MCHR1
SCHEMBL19992536 0.82 TRPA1 (0.44) TRPA1ALDH1A1SMN1; SMN2SLC2A1GABRD
SCHEMBL21182264 0.80 USP7 (0.46) TRPA1ALDH1A1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL21182254 0.80 TRPA1 (0.47) TRPA1CYP11B1CYP11B2MCHR1CYP1A2
SCHEMBL22519104 0.75 ALDH1A1 (0.49) TRPA1ALDH1A1SMN1; SMN2SLC2A1MCHR1
SCHEMBL19992606 0.74 TRPA1 (0.43) TRPA1ALDH1A1SMN1; SMN2SLC2A1CYP11B1
SCHEMBL19992567 0.74 TRPA1 (0.37) TRPA1ALDH1A1SMN1; SMN2SLC2A1CYP11B1
SCHEMBL22303200 0.72 USP7 (0.46) TRPA1ALDH1A1SMN1; SMN2MCHR1USP7
SCHEMBL19992609 0.70 DYRK3 (0.38) TRPA1SMN1; SMN2GABRDGABRB1GABRA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3514155-B1 HETEROCYCLIC COMPOUND, AND HARMFUL-ARTHROPOD-CONTROLLING AGENT CONTAINING SAME SUMITOMO CHEMICAL CO (JP) 2021-06-09 EP disclosed
EP-3514155-A1 HETEROCYCLIC COMPOUND, AND HARMFUL-ARTHROPOD-CONTROLLING AGENT CONTAINING SAME Sumitomo Chemical Company, Limited (JP) 2019-07-24 EP disclosed