SCHEMBL21183104

SCHEMBL21183104

C=CC(=N)Oc1ccc(-c2ccc(OC(=O)C=C)cc2F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.39
SCN9A Q15858 1/20 0.33
GRM2 Q14416 1/20 0.32
ERN1 O75460 1/20 0.32
PRKAB2 O43741 2/20 0.31
PRKAG1 P54619 2/20 0.31
PRKAA2 P54646 2/20 0.31
PRKAA1 Q13131 2/20 0.31
PRKAG3 Q9UGI9 2/20 0.31
PRKAG2 Q9UGJ0 2/20 0.31
PRKAB1 Q9Y478 2/20 0.31
PRKCZ Q05513 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
FFAR4 Q5NUL3 2/20 0.31
APP P05067 1/20 0.30
CYP2C19 P33261 1/20 0.30
GPR35 Q9HC97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9607789 0.91 THRB (0.45) THRBSCN9AGRM2ERN1PRKAB2
SCHEMBL21183107 0.90 THRB (0.38) THRBERN1ESR1ESR2APP
SCHEMBL18432985 0.86 ESR1 (0.34) THRBERN1ESR1ESR2FFAR4
SCHEMBL21475263 0.85 THRB (0.38) THRBESR1ESR2APPCYP2C19
SCHEMBL23045942 0.83 THRB (0.43) THRB
SCHEMBL19157824 0.83 ERN1 (0.46) THRBGRM2ERN1PRKAB2PRKAG1
SCHEMBL18436317 0.82 THRB (0.39) THRBSCN9AGRM2ERN1PRKAB2
SCHEMBL9607903 0.81 THRB (0.44) THRBERN1ESR1ESR2APP
SCHEMBL21592059 0.81 THRB (0.41) THRBCYP2C19
SCHEMBL9607850 0.80 THRB (0.43) THRBERN1ESR1ESR2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3112440-B1 LIQUID-CRYSTAL MEDIUM MERCK PATENT GMBH (DE) 2019-07-24 EP disclosed