SCHEMBL21187121

SCHEMBL21187121

Clc1cccc(N/C(=N\I)NC2CCC(c3ccccc3)CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
LMNA P02545 4/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
EPHX2 P34913 2/20 0.46
EPHX1 P07099 1/20 0.46
TSHR P16473 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
GRIN2B Q13224 1/20 0.46
MAPT P10636 4/20 0.42
HTT P42858 2/20 0.42
THRB P10828 1/20 0.41
CRHR1 P34998 1/20 0.40
TP53 P04637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
RIPK1 Q13546 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17730029 0.81 LMNA (0.70) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL17730073 0.81 LMNA (0.70) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL21187086 0.81 MEN1 (0.49) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL4911807 0.81 LMNA (0.70) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL21187084 0.81 MEN1 (0.49) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL21187213 0.76 NPC1 (0.48) MEN1KMT2ANPC1RAB9AEPHX2
SCHEMBL21187117 0.74 IDO1 (0.51) CYP3A4CYP2C19
SCHEMBL21187139 0.74 NPC1 (0.45) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL21187111 0.74 NPC1 (0.45) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL21187193 0.72 THRB (0.38) NPC1RAB9AEPHX2EPHX1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed