SCHEMBL21187158

SCHEMBL21187158

C/N=C(\Nc1ccc(OC)c(F)c1)NC1CCC(c2ccnc(C)c2F)CC1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.37
PDE4D Q08499 1/20 0.37
AXL P30530 5/20 0.36
CASP3 P42574 1/20 0.35
CDK9 P50750 1/20 0.35
CASP7 P55210 1/20 0.35
MET P08581 10/20 0.35
MAP2K1 Q02750 1/20 0.34
SLC11A2 P49281 1/20 0.34
KDR P35968 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187092 0.87 EPHX2 (0.38) MET
SCHEMBL21187154 0.84 NPC1 (0.36) METKDR
SCHEMBL21187097 0.82 IDO1 (0.40)
SCHEMBL21187096 0.81 MEN1 (0.39) KDR
SCHEMBL21187168 0.79 GRM4 (0.41) PDE4BPDE4DCASP3CDK9CASP7
SCHEMBL21187166 0.79 MET (0.37) PDE4BPDE4DAXLCASP3CDK9
SCHEMBL21187159 0.76 IDO1 (0.37) METKDR
SCHEMBL21187156 0.72 NPC1 (0.43) CASP3
SCHEMBL21187221 0.70 IDO1 (0.39) MET
SCHEMBL21187219 0.68 CHRM4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed