SCHEMBL21187168

SCHEMBL21187168

COc1cc(NC(=N)NC2CCC(c3ccnc(C)c3F)CC2)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 2/20 0.41
PDE4B Q07343 2/20 0.38
CASP3 P42574 1/20 0.36
CDK9 P50750 1/20 0.36
CASP7 P55210 1/20 0.36
CYP17A1 P05093 1/20 0.35
RAB9A P51151 1/20 0.34
MET P08581 1/20 0.34
FGFR4 P22455 1/20 0.34
IDO1 P14902 4/20 0.34
KCNH2 Q12809 2/20 0.34
KDR P35968 2/20 0.34
HRH2 P25021 1/20 0.34
TRPC5 Q9UL62 1/20 0.34
BRAF P15056 2/20 0.33
RAF1 P04049 1/20 0.33
CYP2C9 P11712 2/20 0.33
TGFBR1 P36897 1/20 0.33
PDE4D Q08499 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187166 0.85 MET (0.37) PDE4BCASP3CDK9CASP7MET
SCHEMBL21187156 0.85 NPC1 (0.43) GRM4CASP3RAB9A
SCHEMBL21187221 0.84 IDO1 (0.39) RAB9AMETIDO1KCNH2CYP2C9
SCHEMBL21187158 0.79 PDE4B (0.37) PDE4BCASP3CDK9CASP7MET
SCHEMBL21187153 0.74 NPC1 (0.45) GRM4CASP3RAB9A
SCHEMBL21187157 0.74 NPC1 (0.41) RAB9AIDO1
SCHEMBL21187146 0.74 SMN1; SMN2 (0.41) CYP2C9
SCHEMBL21187131 0.73 IDO1 (0.50) RAB9AIDO1KCNH2KDRCYP2C9
SCHEMBL21187138 0.73 IDO1 (0.50) RAB9AIDO1KCNH2KDRCYP2C9
SCHEMBL21187092 0.73 EPHX2 (0.38) RAB9AMETIDO1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed