SCHEMBL21187236

SCHEMBL21187236

C=C1CNCC(Cc2cccc(CCCc3ccc(CC)cc3)c2)N1

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.32
PDE4A P27815 2/20 0.31
MAPK1 P28482 2/20 0.31
PDE4D Q08499 2/20 0.31
TNF P01375 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
NFKB1 P19838 1/20 0.31
KMT2A Q03164 1/20 0.31
CXCR4 P61073 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187235 0.86 CXCR4 (0.39) HTR2APDE4AMAPK1PDE4DTNF
SCHEMBL28225986 0.86 CXCR4 (0.39) HTR2APDE4AMAPK1PDE4DTNF
SCHEMBL29452904 0.86 CXCR4 (0.39) HTR2APDE4AMAPK1PDE4DTNF
SCHEMBL28225984 0.86 CXCR4 (0.39) HTR2APDE4AMAPK1PDE4DTNF
SCHEMBL28226022 0.79 HRH3 (0.40) HTR2A
SCHEMBL28226023 0.79 HRH3 (0.40) HTR2A
SCHEMBL13427805 0.74 MEN1 (0.42) MEN1KMT2A
SCHEMBL21187254 0.74 SIGMAR1 (0.33) HTR2A
SCHEMBL21176956 0.72 POLB (0.55) KMT2A
SCHEMBL28225275 0.71 CYP2D6 (0.36) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed