SCHEMBL21187254

SCHEMBL21187254

C=C1CN(C)C(Cc2cccc(CCCc3ccc(CC)cc3)c2)N1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.33
HTR2A P28223 1/20 0.32
OPRM1 P35372 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22555679 0.86 OPRK1 (0.36) SIGMAR1HTR2AALDH1A1
SCHEMBL30514796 0.86 OPRK1 (0.36) SIGMAR1HTR2AALDH1A1
SCHEMBL21187251 0.86 OPRK1 (0.36) SIGMAR1HTR2AALDH1A1
SCHEMBL21187236 0.74 HTR2A (0.32) HTR2A
SCHEMBL28225275 0.71 CYP2D6 (0.36) SIGMAR1HTR2ATAAR1
SCHEMBL29452916 0.68 GPR84 (0.34) HTR2A
SCHEMBL21176974 0.68 GPR84 (0.34) HTR2A
SCHEMBL21176977 0.68 GPR84 (0.34) HTR2A
SCHEMBL21176956 0.67 POLB (0.55) SLC6A2SLC6A4SLC6A3
SCHEMBL28226022 0.67 HRH3 (0.40) SIGMAR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed