SCHEMBL21187280

SCHEMBL21187280

I[C@H]1CC[C@@H](Oc2cc(N3CCOCC3)cc3c2CCCCCN3)CC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 16/20 0.33
IKBKE Q14164 2/20 0.33
SYK P43405 1/20 0.31
TTK P33981 1/20 0.30
LRRK2 Q5S007 1/20 0.30
NQO1 P15559 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187323 0.81 TTK (0.34) TTK
SCHEMBL21187279 0.74 PRKDC (0.39) NQO1
SCHEMBL21187390 0.74 MAPT (0.35) NQO1
SCHEMBL21187388 0.71 FLT3 (0.35) SYKTTK
SCHEMBL23059584 0.61
SCHEMBL21187792 0.61
SCHEMBL21286545 0.61
SCHEMBL20216508 0.61
SCHEMBL16038633 0.59 SYK (0.43) TBK1IKBKESYKLRRK2
SCHEMBL16040024 0.59 SYK (0.43) TBK1IKBKESYKLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143678-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-07-25 WO disclosed