SCHEMBL21188481

SCHEMBL21188481

Cc1noc(C)c1-c1ccc(C=N)c(N)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.44
BRD2 P25440 1/20 0.40
JAK2 O60674 1/20 0.39
MBOAT4 Q96T53 1/20 0.39
TLR8 Q9NR97 1/20 0.39
CYP1A2 P05177 6/20 0.38
CYP3A4 P08684 4/20 0.38
USP2 O75604 2/20 0.38
TDO2 P48775 1/20 0.38
ERN1 O75460 2/20 0.37
CREBBP Q92793 1/20 0.37
CLK4 Q9HAZ1 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
HIF1A Q16665 1/20 0.36
AURKA O14965 3/20 0.36
AURKB Q96GD4 3/20 0.36
CYP2C19 P33261 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17875696 0.81 BRD4 (0.44) BRD4BRD2JAK2MBOAT4TLR8
SCHEMBL21188508 0.77 BRD4 (0.39) BRD4BRD2JAK2MBOAT4TLR8
SCHEMBL18319367 0.72 ERN1 (0.43) BRD4BRD2JAK2MBOAT4TLR8
SCHEMBL19296089 0.70 BRD4 (0.44) BRD4BRD2CYP1A2CYP3A4USP2
SCHEMBL17875699 0.70 BRD4 (0.40) BRD4BRD2CYP1A2CYP3A4USP2
SCHEMBL30522617 0.69 BRD4 (0.46) BRD4BRD2JAK2TLR8CYP1A2
SCHEMBL29836739 0.69 BRD4 (0.46) BRD4BRD2JAK2MBOAT4TLR8
SCHEMBL14620954 0.69 KDM4E (0.44) TLR8CYP1A2USP2ALDH1A1KMT2A
SCHEMBL17643820 0.69 BRD4 (0.40) BRD4BRD2CYP1A2CYP3A4USP2
SCHEMBL4102764 0.68 TLR8 (0.40) BRD4BRD2JAK2MBOAT4TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143719-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) SYROS PHARMACEUTICALS, INC. (US) 2019-07-25 WO disclosed