SCHEMBL21188508

SCHEMBL21188508

CC(=N)c1ccc(-c2c(C)noc2C)nc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.39
BRD2 P25440 2/20 0.38
MBOAT4 Q96T53 1/20 0.37
JAK2 O60674 1/20 0.37
TLR8 Q9NR97 1/20 0.37
CYP1A2 P05177 4/20 0.37
CYP3A4 P08684 2/20 0.37
USP2 O75604 1/20 0.37
CREBBP Q92793 1/20 0.36
AR P10275 1/20 0.35
AURKA O14965 3/20 0.35
AURKB Q96GD4 3/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
MLYCD O95822 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17875696 0.79 BRD4 (0.44) BRD4BRD2MBOAT4JAK2TLR8
SCHEMBL21188481 0.77 BRD4 (0.44) BRD4BRD2MBOAT4JAK2TLR8
SCHEMBL21188151 0.74 CCNT1 (0.35) BRD4CYP1A2CYP3A4USP2AURKA
SCHEMBL21188480 0.71 PDE5A (0.35) BRD4BRD2CYP1A2CYP3A4AURKA
SCHEMBL18319367 0.70 ERN1 (0.43) BRD4BRD2MBOAT4JAK2TLR8
SCHEMBL29836739 0.67 BRD4 (0.46) BRD4BRD2MBOAT4JAK2TLR8
SCHEMBL30522617 0.67 BRD4 (0.46) BRD4BRD2JAK2TLR8CYP1A2
SCHEMBL19057174 0.67 FGFR1 (0.42) ALDH1A1
SCHEMBL12270079 0.65 CCR1 (0.54) BRD4BRD2MBOAT4CYP1A2CYP3A4
SCHEMBL17875697 0.65 ALDH1A1 (0.39) BRD4BRD2MBOAT4JAK2TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143719-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) SYROS PHARMACEUTICALS, INC. (US) 2019-07-25 WO disclosed