SCHEMBL21189608

SCHEMBL21189608

CCOC(=O)c1cc(Cl)n2nc(C)c(C)c2n1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
ADORA2A P29274 1/20 0.41
ADORA3 P0DMS8 2/20 0.41
MAPT P10636 1/20 0.40
POLB P06746 2/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
LMNA P02545 1/20 0.39
NOTUM Q6P988 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177528 0.88 ADORA3 (0.42) CYP1A2ADORA2AADORA3MAPTPOLB
SCHEMBL21177355 0.87 ADORA3 (0.42) CYP1A2ADORA2AADORA3MAPTPOLB
SCHEMBL20064665 0.86 CYP1A2 (0.44) CYP1A2ADORA2AADORA3MAPTPOLB
SCHEMBL20723167 0.82 CYP1A2 (0.45) CYP1A2ADORA2AMAPTKDM4EALDH1A1
SCHEMBL25465499 0.81 MAPT (0.38) MAPTPOLBKDM4EALDH1A1HPGD
SCHEMBL21189850 0.79 KDM4E (0.45) CYP1A2MAPTPOLBKDM4EALDH1A1
SCHEMBL20568880 0.78 GSK3B (0.45) CYP1A2ADORA2AMAPTPOLBKDM4E
SCHEMBL9679448 0.78 ALDH1A1 (0.48) CYP1A2ADORA2AADORA3POLBKDM4E
SCHEMBL21177423 0.77 KDM4E (0.45) CYP1A2ADORA2AMAPTPOLBKDM4E
SCHEMBL20568271 0.76 GSK3B (0.44) CYP1A2ADORA2AMAPTPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141694-A1 PI4KIIIBETA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-07-25 WO disclosed