SCHEMBL21189732

SCHEMBL21189732

CN(CCO)C(=O)c1cc(B2OC(C)(C)C(C)(C)O2)ccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LIPG Q9Y5X9 3/20 0.35
ROCK1 Q13464 1/20 0.34
LPL P06858 2/20 0.34
PDK2 Q15119 1/20 0.34
HIF1A Q16665 3/20 0.34
F11 P03951 2/20 0.33
MAPT P10636 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
P4HB P07237 1/20 0.33
LRRK2 Q5S007 1/20 0.32
HDAC4 P56524 1/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
P2RX7 Q99572 1/20 0.32
F2 P00734 1/20 0.32
PRSS1 P07477 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177337 0.93 PDK2 (0.36) AAK1ALDH1A1LIPGROCK1LPL
SCHEMBL21179344 0.86 HIF1A (0.36) ALDH1A1LIPGROCK1LPLHIF1A
SCHEMBL22858943 0.86 HIF1A (0.36) AAK1ALDH1A1LIPGROCK1LPL
SCHEMBL21177390 0.86 TSHR (0.38) AAK1ALDH1A1LIPGROCK1LPL
SCHEMBL21177403 0.83 CSF1R (0.38) AAK1LIPGROCK1HIF1ALRRK2
SCHEMBL24108583 0.83 ALDH1A1 (0.40) AAK1ALDH1A1LIPGROCK1LPL
SCHEMBL21179433 0.80 HIF1A (0.35) LIPGROCK1LPLPDK2HIF1A
SCHEMBL22922489 0.79 HDAC4 (0.43) LIPGLPLPDK2F11CA1
SCHEMBL18274838 0.78 LPL (0.48) LIPGLPL
SCHEMBL1721722 0.77 ALDH1A1 (0.47) AAK1ALDH1A1LIPGROCK1LPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117069728-A PI4KIII beta inhibitors 葛兰素史克知识产权开发有限公司 2023-11-17 CN disclosed
CN-111868063-A PI4KIII beta inhibitors 葛兰素史克知识产权开发有限公司 2020-10-30 CN disclosed
WO-2019141694-A1 PI4KIIIBETA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-07-25 WO disclosed