SCHEMBL21190885

SCHEMBL21190885

CNS(=O)(=O)c1ccc(Oc2ccc(F)cc2)c(Br)c1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
EPAS1 Q99814 13/20 0.51
BRD4 O60885 1/20 0.50
SLC6A4 P31645 2/20 0.47
SOS1 Q07889 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
HTR2A P28223 1/20 0.45
KCNH2 Q12809 1/20 0.45
SCN9A Q15858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24631128 0.86 SOS1 (0.50) LMNAHTTSMN1; SMN2EPAS1SLC6A4
SCHEMBL24631132 0.86 CA12 (0.54) LMNAHTTSMN1; SMN2EPAS1SLC6A4
SCHEMBL24631317 0.85 LMNA (0.49) LMNAHTTSMN1; SMN2EPAS1BRD4
SCHEMBL24631133 0.85 EPAS1 (0.50) LMNAHTTSMN1; SMN2EPAS1SLC6A4
SCHEMBL24631315 0.84 LMNA (0.50) LMNAHTTSMN1; SMN2EPAS1BRD4
SCHEMBL24631135 0.83 ALDH1A1 (0.50) LMNAHTTSMN1; SMN2EPAS1SLC6A4
SCHEMBL28750635 0.80 SMN1; SMN2 (0.81) LMNAHTTSMN1; SMN2SOS1
SCHEMBL1471508 0.80 FFAR4 (0.60) LMNA
SCHEMBL4926851 0.77 POLB (0.62) LMNAHTTSMN1; SMN2
SCHEMBL22718133 0.77 EPAS1 (0.50) EPAS1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022177869-A1 ARYL ETHER COMPOUNDS AS TEAD MODULATORS MERCK SHARP & DOHME LLC (US) 2022-08-25 WO disclosed
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed