Corydalmine

Corydalmine

SCHEMBL21192512

COc1cc2c(cc1OC)[C@@H]1Cc3ccc(O)c(OC)c3CN1CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 16/20 1.00
DRD2 P14416 13/20 1.00
DRD3 P35462 9/20 1.00
F3 P13726 6/20 1.00
DRD5 P21918 5/20 1.00
HTR1A P08908 1/20 1.00
SIGMAR1 Q99720 3/20 0.89
DRD4 P21917 2/20 0.89
ADRA1D P25100 1/20 0.89
ADRA1A P35348 1/20 0.89
ADRA1B P35368 1/20 0.89
CYP3A4 P08684 1/20 0.80
LMNA P02545 1/20 0.79
TSHR P16473 1/20 0.79
ACHE P22303 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Corydalmine SCHEMBL12667453 1.00 DRD1 (1.00) DRD1DRD2DRD3F3DRD5
Corydalmine SCHEMBL29243055 0.99 DRD1 (0.98) DRD1DRD2DRD3F3DRD5
Stepholidine SCHEMBL29943869 0.94 DRD1 (1.00) DRD1DRD2DRD3F3DRD5
Stepholidine SCHEMBL460434 0.94 DRD1 (1.00) DRD1DRD2DRD3F3DRD5
Stepholidine SCHEMBL10001966 0.94 DRD1 (1.00) DRD1DRD2DRD3F3DRD5
Stepholidine SCHEMBL10001965 0.94 DRD1 (1.00) DRD1DRD2DRD3F3DRD5
Stepholidine SCHEMBL29414100 0.94 DRD1 (1.00) DRD1DRD2DRD3F3DRD5
SCHEMBL26326556 0.92 DRD1 (0.85) DRD1DRD2DRD3F3DRD5
SCHEMBL22057260 0.91 DRD1 (0.83) DRD1DRD2DRD3F3DRD5
Demethylcorydalmine SCHEMBL12943247 0.89 DRD1 (0.84) DRD1DRD2DRD3F3DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112812112-B Preparation method of isoquinoline alkaloid L-corydaline 杨征 2024-06-28 CN disclosed
EP-3517537-B1 DEUTERATED DERIVATIVE OF L-TETRAHYDROPALMATINE AND MEDICAL USE THEREOF TAIZHOU HUAYUAN MEDICINAL TECH CO LTD (CN) 2023-09-13 EP disclosed
EP-3517537-B1 DEUTERATED DERIVATIVE OF L-TETRAHYDROPALMATINE AND MEDICAL USE THEREOF TAIZHOU HUAYUAN MEDICINAL TECH CO LTD (CN) 2023-09-13 EP disclosed
US-11236081-B2 Crystalline salts of corydalmine Yang, Zheng (CN) 2022-02-01 US disclosed
US-20210347770-A1 CRYSTALLINE SALTS OF CORYDALMINE YANG, ZHENG (CN) 2021-11-11 US disclosed
WO-2020107335-A1 CRYSTALLINE SALTS OF CORYDALMINE YANG ZHENG (CN) 2020-06-04 WO disclosed
WO-2020108330-A1 CRYSTALLINE SALTS OF CORYDALMINE YANG ZHENG (CN) 2020-06-04 WO disclosed
US-10617679-B2 Deuterated compounds and medical uses thereof JINGLUWEIDAI INFORMATION CONSULTING SERVICE (BEIJING) CO. LTD. (CN) 2020-04-14 US disclosed
US-10617679-B2 Deuterated compounds and medical uses thereof JINGLUWEIDAI INFORMATION CONSULTING SERVICE (BEIJING) CO. LTD. (CN) 2020-04-14 US disclosed
US-20190240204-A1 DEUTERATED COMPOUNDS AND MEDICAL USES THEREOF TAIZHOU HUAYUAN MEDICINAL TECH CO. LTD. (CN) 2019-08-08 US disclosed
US-20190240204-A1 DEUTERATED COMPOUNDS AND MEDICAL USES THEREOF TAIZHOU HUAYUAN MEDICINAL TECH CO. LTD. (CN) 2019-08-08 US disclosed
EP-3517537-A1 DEUTERATED DERIVATIVE OF L-TETRAHYDROPALMATINE AND MEDICAL USE THEREOF Jingluweidai Information Consulting Service (Beijing) Co Ltd (CN) 2019-07-31 EP disclosed
EP-3517537-A1 DEUTERATED DERIVATIVE OF L-TETRAHYDROPALMATINE AND MEDICAL USE THEREOF Jingluweidai Information Consulting Service (Beijing) Co Ltd (CN) 2019-07-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10617679-B2 Deuterated compounds and medical uses thereof HRH4, HRH3, LPAR3 DRD1 251/4885DRD2 213/4885DRD3 154/4885
US-20190240204-A1 DEUTERATED COMPOUNDS AND MEDICAL USES THEREOF HRH4, HRH3, LPAR3 DRD1 251/4885DRD2 213/4885DRD3 154/4885
US-20210347770-A1 CRYSTALLINE SALTS OF CORYDALMINE NPC1L1, CHLSN, LIPA DRD1 37/4885DRD2 50/4885DRD3 133/4885
US-11236081-B2 Crystalline salts of corydalmine NPC1L1, CHLSN, LIPA DRD1 37/4885DRD2 50/4885DRD3 133/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.