SCHEMBL21202802

SCHEMBL21202802

CC(C)(O)C(C)(C)OBc1ccc(-n2c(-c3cc(-c4nc5ccccc5n4-c4ccc(B5OC(C)(C)C(C)(C)O5)cc4)cc(-c4nc5ccccc5n4-c4ccc(B5OC(C)(C)C(C)(C)O5)cc4)c3)nc3ccccc32)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 5/20 0.39
ESR1 P03372 4/20 0.39
GRIA1 P42261 1/20 0.36
CACNG8 Q8WXS5 1/20 0.36
CACNG2 Q9Y698 1/20 0.36
LPL P06858 2/20 0.35
LIPG Q9Y5X9 2/20 0.35
HDAC1 Q13547 3/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
SNCA P37840 1/20 0.33
RPS6KB1 P23443 1/20 0.33
ROCK1 Q13464 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
PTGS2 P35354 1/20 0.32
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18015678 0.85 ESR2 (0.48) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL18597398 0.82 ESR2 (0.57) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL17536059 0.80 ESR1 (0.51) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL15336505 0.79 ESR1 (0.50) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL29603396 0.79 ESR2 (0.58) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL12424886 0.79 ESR2 (0.58) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL15770520 0.78 ESR1 (0.47) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL14854199 0.78 CA1 (0.43) ESR2LPLLIPGSNCACA1
SCHEMBL25875540 0.77 ESR2 (0.51) ESR2ESR1GRIA1CACNG8CACNG2
SCHEMBL19193834 0.77 LIPG (0.57) ESR2ESR1GRIA1CACNG8CACNG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3254317-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-07-31 EP disclosed