Dimethyl Fumarate

Dimethyl Fumarate

SCHEMBL21219085

COC(=O)/C=C/C(=O)OC.N

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Dimethyl Fumarate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.93
NFE2L2 Q16236 3/20 0.93
HCAR2 Q8TDS4 2/20 0.93
ALDH1A1 P00352 7/20 0.46
MAPT P10636 5/20 0.46
KDM4E B2RXH2 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
TYR P14679 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
GFPT1 Q06210 1/20 0.43
ALOX15 P16050 2/20 0.43
HSD17B10 Q99714 2/20 0.43
RECQL P46063 1/20 0.43
TTR P02766 1/20 0.40
APP P05067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethyl Maleate SCHEMBL15902274 1.00 NFE2L2 (0.93) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Fumarate SCHEMBL28128958 0.96 NFE2L2 (1.00) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Maleate SCHEMBL27720952 0.96 NFE2L2 (1.00) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Fumarate SCHEMBL41836 0.96 NFE2L2 (1.00) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Maleate SCHEMBL75864 0.96 NFE2L2 (1.00) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Fumarate SCHEMBL41835 0.96 NFE2L2 (1.00) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Fumarate SCHEMBL11668350 0.96 NFE2L2 (1.00) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Maleate SCHEMBL28991725 0.93 NFE2L2 (0.93) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Maleate SCHEMBL7057632 0.93 HCAR2 (0.93) NFE2L2HCAR2KEAP1ALDH1A1MAPT
Dimethyl Fumarate SCHEMBL29395244 0.93 NFE2L2 (0.93) NFE2L2HCAR2KEAP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3518878-A1 IMPROVED CONDITIONING HAIR TREATMENT PRODUCT WITH WASHOUT PROTECTION Henkel AG & Co. KGaA (DE) 2019-08-07 EP disclosed