SCHEMBL21233337

SCHEMBL21233337

Cc1c(-c2ccccn2)cnn1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.47
ALDH1A1 P00352 3/20 0.47
LMNA P02545 3/20 0.46
CCR1 P32246 2/20 0.46
CCR5 P51681 2/20 0.46
CCR8 P51685 2/20 0.46
POLB P06746 2/20 0.46
HIF1A Q16665 2/20 0.46
CYP1A2 P05177 1/20 0.46
METAP1 P53582 1/20 0.46
BLM P54132 1/20 0.46
DOHH Q9BU89 1/20 0.46
P4HTM Q9NXG6 1/20 0.46
BRD4 O60885 2/20 0.46
CYP11B2 P19099 1/20 0.44
CREBBP Q92793 1/20 0.43
TP53 P04637 4/20 0.43
NPC1 O15118 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10559743 0.84 BRD4 (0.45) KDM4EALDH1A1LMNACCR1CCR5
SCHEMBL10561671 0.82 PIM1 (0.46) KDM4EALDH1A1LMNACCR1CCR5
SCHEMBL10520969 0.82 TDO2 (0.47) KDM4EALDH1A1LMNACCR1CCR5
SCHEMBL30674979 0.82 BRD4 (0.51) KDM4ELMNACCR1CCR5CCR8
SCHEMBL15345069 0.80 CCR1 (0.55) KDM4EALDH1A1CCR1CCR5CCR8
SCHEMBL8138943 0.80 KDR (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL22952795 0.80 BRD4 (0.42) KDM4EALDH1A1LMNACCR1CCR5
SCHEMBL21233353 0.79 BRD4 (0.44) KDM4EALDH1A1POLBBRD4CYP11B2
SCHEMBL21233352 0.79 CYP11B2 (0.43) KDM4EALDH1A1POLBHIF1ABLM
SCHEMBL21233346 0.78 BRD4 (0.43) KDM4EALDH1A1POLBCYP1A2BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019148851-A1 FIVE-MEMBERED RING-SUBSTITUTED PYRIDAZINOL COMPOUND AND DERIVATIVES THEREOF, PREPARATION METHOD, HERBICIDAL COMPOSITION, AND APPLICATION 青岛清原化合物有限公司 2019-08-08 WO disclosed
WO-2019149260-A1 PYRIDAZINOL COMPOUND, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, HERBICIDAL COMPOSITION AND USE THEREOF 青岛清原化合物有限公司 2019-08-08 WO disclosed