SCHEMBL21236877

SCHEMBL21236877

Cc1cc(NCc2cccnc2)cc(-c2ccc(Oc3ccc(F)cc3)cc2)n1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 6/20 0.71
CYP3A4 P08684 6/20 0.53
CYP2C9 P11712 6/20 0.53
CYP2C19 P33261 6/20 0.53
CYP2D6 P10635 3/20 0.53
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 3/20 0.51
CYP1A2 P05177 2/20 0.51
HSD17B10 Q99714 2/20 0.48
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NOS2 P35228 1/20 0.47
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
PABPC1 P11940 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29421458 0.83 SCN9A (1.00) SCN9A
SCHEMBL787412 0.83 SCN9A (1.00) SCN9A
SCHEMBL24517122 0.82 SCN9A (0.62) SCN9ACYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL13270542 0.76 SCN9A (0.51) SCN9A
SCHEMBL22530412 0.75 SCN9A (0.55) SCN9ACYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL22530411 0.74 ALDH1A1 (0.55) SCN9ACYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL22530931 0.73 ALDH1A1 (0.63) SCN9ACYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL10371775 0.72 LTA4H (0.72) CYP3A4CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL22530439 0.71 CYP3A4 (0.56) SCN9ACYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL22531085 0.71 ALDH1A1 (0.49) SCN9ACYP3A4CYP2C9CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616441-B1 PYRIDINE COMPOUNDS AND THE USES THEREOF PURDUE PHARMA LP (US) 2019-08-07 EP disclosed