SCHEMBL21242580

SCHEMBL21242580

O=C(NC1CCC(c2cccc3nc(NC(O)C4CC4)nn23)CC1)[C@@H]1CC1(F)F

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 20/20 0.73
TYK2 P29597 20/20 0.73
JAK2 O60674 19/20 0.73
JAK3 P52333 14/20 0.73
CYP2C19 P33261 3/20 0.73
CYP1A2 P05177 1/20 0.73
CYP2C9 P11712 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23080443 0.84 JAK1 (1.00) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL21242563 0.84 JAK1 (1.00) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL21242552 0.84 JAK1 (1.00) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL21242564 0.84 JAK1 (1.00) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL24742801 0.81 JAK2 (0.73) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL24742806 0.71 JAK2 (0.69) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL23424241 0.71 JAK2 (0.69) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL21757167 0.71 JAK2 (0.69) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL21242553 0.71 JAK2 (1.00) JAK1TYK2JAK2JAK3CYP2C19
SCHEMBL24653307 0.71 JAK2 (0.68) JAK1TYK2JAK2JAK3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019149244-A1 JAK INHIBITOR AND USE THEREOF 南京明德新药研发股份有限公司 2019-08-08 WO disclosed