SCHEMBL21243066

SCHEMBL21243066

CCOC(=O)CC(C(=O)c1ccc2ccc(C)cc2c1)c1ccncc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
NAMPT P43490 1/20 0.36
SYK P43405 1/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
ROCK2 O75116 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
RAPGEF3 O95398 1/20 0.32
ELANE P08246 1/20 0.32
HSD17B14 Q9BPX1 1/20 0.31
MAPK1 P28482 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16061977 0.91 CCNC (0.40) NAMPTHPGDKDM4EALDH1A1GAA
SCHEMBL23587032 0.83 CYP2A6 (0.42) CYP2A6NAMPTHSD17B10HPGDALDH1A1
SCHEMBL16092088 0.76 CDC25B (0.43) HPGDKDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL5847575 0.73 SMN1; SMN2 (0.46) NAMPTHPGDKDM4EALDH1A1GAA
SCHEMBL14523452 0.69 MAPT (0.42) KDM4EALDH1A1CASP1SMN1; SMN2NPC1
SCHEMBL4672007 0.68 LTA4H (0.42) NAMPTNPC1MAPT
SCHEMBL26933366 0.66 ROCK2 (0.37) NAMPTHSD17B10HPGDKDM4EALDH1A1
SCHEMBL15704203 0.66 CYP2A6 (0.61) CYP2A6HSD17B10HPGDKDM4EALDH1A1
SCHEMBL12600053 0.65 HDAC3 (0.48) NAMPTKDM4EALDH1A1SMN1; SMN2NPC1
SCHEMBL17736033 0.65 SLC6A2 (0.47) HPGDKDM4EALDH1A1GAAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3842424-A1 MAP KINASE MODULATORS AND USES THEREOF IN THE TRETAMENT OF TAUOPATHIES The Trustees of Columbia University in the City of New York (US) 2021-06-30 EP disclosed
EP-3521284-A1 PYRAZINE COMPOUNDS AS MAP KINASE MODULATORS AND USES THEREOF The Trustees of Columbia University in the City of New York (US) 2019-08-07 EP disclosed