SCHEMBL2124455

SCHEMBL2124455

N=C(N)c1cncc2c1ccn2O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3752264 0.75 F10 (0.33)
SCHEMBL16897117 0.66 PARP1 (0.33)
Hydrochloric Acid SCHEMBL20270500 0.64 PRKCZ (0.42)
SCHEMBL2126361 0.63 F2 (0.39)
SCHEMBL17654485 0.61 PLAU (0.61)
SCHEMBL12067334 0.60 EPHB3 (0.45)
Hydrochloric Acid SCHEMBL23754646 0.59 TUBB4A (0.45)
Hydrochloric Acid SCHEMBL1693996 0.59 EPHB3 (0.44)
SCHEMBL7958530 0.58 GAA (0.45)
SCHEMBL1421583 0.58 SIRT3 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443115-A1 COMPOUNDS Glaxo Group Limited (GB) 2012-04-25 EP disclosed
WO-2010145201-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed