SCHEMBL21254007

SCHEMBL21254007

NC(=O)C[C@H](NC(=O)CCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.54
ACE P12821 1/20 0.51
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.46
RAB9A P51151 1/20 0.46
GLS O94925 1/20 0.46
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
MBTPS1 Q14703 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30910805 0.88 ACE (0.50) CASP1ACEPOLBALDH1A1RAB9A
SCHEMBL18812968 0.86 CASP1 (0.50) CASP1ACEALDH1A1GLSHDAC2
SCHEMBL11940461 0.85 POLB (0.51) CASP1ACEPOLBALDH1A1RAB9A
SCHEMBL28252941 0.85 EPHX2 (0.50) ACE
SCHEMBL28252940 0.85 EPHX2 (0.50) ACE
SCHEMBL13673884 0.85 ACE (0.67) CASP1ACEPOLBALDH1A1HDAC8
SCHEMBL4152421 0.85 ACE (0.67) CASP1ACEPOLBALDH1A1HDAC8
SCHEMBL16908006 0.85 HDAC2 (0.51) ALDH1A1RAB9AHDAC2HDAC8HDAC6
SCHEMBL28680572 0.85 ALDH1A1 (0.58) ACEALDH1A1RAB9AHDAC2HDAC8
SCHEMBL5272643 0.85 ALDH1A1 (0.58) ACEALDH1A1RAB9AHDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092244-B1 DIPEPTIDES AS INHIBITORS OF HUMAN IMMUNOPROTEASOMES UNIV CORNELL (US) 2019-08-14 EP disclosed