SCHEMBL21254504

SCHEMBL21254504

c1ccc(CN2CCOC3(CCOCC3)C2)cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 4/20 0.57
CHRM2 P08172 2/20 0.47
CHRM3 P20309 2/20 0.47
SIGMAR1 Q99720 4/20 0.47
OPRM1 P35372 1/20 0.47
CYP3A4 P08684 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
CYP2D6 P10635 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26552039 0.92 MGLL (0.60) MGLLCHRM2CHRM3SIGMAR1OPRM1
SCHEMBL21254493 0.89 MGLL (0.58) MGLLCHRM2CHRM3SIGMAR1OPRM1
SCHEMBL18785020 0.87 MGLL (0.56) MGLLCHRM2CHRM3SIGMAR1OPRM1
SCHEMBL18719631 0.85 MGLL (0.58) MGLLCHRM2CHRM3SIGMAR1OPRM1
SCHEMBL20046098 0.85 CYP2D6 (0.58) MGLLCHRM2CHRM3SIGMAR1OPRM1
Hydrochloric Acid SCHEMBL31716831 0.84 CYP2D6 (0.57) MGLLCHRM2CHRM3SIGMAR1OPRM1
SCHEMBL17318952 0.83 SIGMAR1 (0.58) MGLLCHRM2SIGMAR1OPRM1CYP2D6
SCHEMBL17319038 0.82 MGLL (0.70) MGLLCHRM2CHRM3SIGMAR1OPRM1
SCHEMBL21254338 0.82 MGLL (0.55) MGLLCHRM2CHRM3SIGMAR1OPRM1
Hydrochloric Acid SCHEMBL18695858 0.82 SIGMAR1 (0.57) MGLLCHRM2SIGMAR1OPRM1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3113780-B1 HIV PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2019-08-14 EP disclosed