SCHEMBL2126344

SCHEMBL2126344

Oc1nnc(Cl)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GOT1 P17174 1/20 0.50
MAPT P10636 8/20 0.46
ALDH1A1 P00352 6/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
GFER P55789 1/20 0.46
KDM4E B2RXH2 3/20 0.42
RAB9A P51151 4/20 0.40
LMNA P02545 3/20 0.40
POLB P06746 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
NPC1 O15118 3/20 0.38
HTT P42858 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL345211 0.84 GOT1 (0.62) GOT1MAPTALDH1A1SMN1; SMN2HPGD
SCHEMBL30082487 0.84 IDO1 (0.47) MAPTALDH1A1SMN1; SMN2HPGDMEN1
SCHEMBL350637 0.84 IDO1 (0.47) MAPTALDH1A1SMN1; SMN2HPGDMEN1
SCHEMBL29365992 0.84 GOT1 (0.62) GOT1MAPTALDH1A1SMN1; SMN2HPGD
SCHEMBL27758703 0.82 GOT1 (0.60) GOT1MAPTALDH1A1SMN1; SMN2HPGD
Hydrazine SCHEMBL10949625 0.79 KDM4E (0.46) MAPTALDH1A1SMN1; SMN2HPGDMEN1
Bicarbonate SCHEMBL11022555 0.78 GOT1 (0.52) GOT1MAPTALDH1A1SMN1; SMN2HPGD
SCHEMBL31617120 0.76 PDE5A (0.38) MAPTALDH1A1SMN1; SMN2HPGDMEN1
SCHEMBL10906806 0.74 GOT1 (0.48) GOT1MAPTALDH1A1SMN1; SMN2HPGD
SCHEMBL25254434 0.74 EP300 (0.40) MAPTKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190298717-A1 Hydralazine and Active Derivatives Thereof for Neuronal Cell Survival and Regeneration UNIV TEXAS (US) 2019-10-03 US claimed
WO-2017160864-A1 HYDRALAZINE AND ACTIVE DERIVATIVES THEREOF FOR NEURONAL CELL SURVIVAL AND REGENERATION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-09-21 WO claimed
EP-4735433-A2 SUBSTITUTED PYRIDAZINE COMPOUNDS AS INHIBITORS OF NLRP3 ACTIVITY AND THERAPEUTIC USES THEREOF Viva Star Biosciences (US) Inc. (US) 2026-05-06 EP disclosed
WO-2025006681-A2 SUBSTITUTED PYRIDAZINE COMPOUNDS AS INHIBITORS OF NLRP3 ACTIVITY AND THERAPEUTIC USES THEREOF VIVA STAR BIOSCIENCES (US) INC. (US) 2025-01-02 WO disclosed
EP-3189049-B1 PHTHALAZINE DERIVATIVES OF FORMULA (I) AS PCAF AND GCN5 INHIBITORS FOR USE IN THE TREATMENT OF CANCER GENENTECH INC (US) 2024-03-20 EP disclosed
CN-117659025-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-03-08 CN disclosed
CN-117586108-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN disclosed
CN-117586191-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN disclosed
CN-111542515-B TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2023-12-05 CN disclosed
US-20230132035-A1 Toll-Like Receptor 8 (TLR8)-Specific Antagonists and Methods of Making and Uses Thereof UNIV COLORADO REGENTS (US) 2023-04-27 US disclosed
US-11466010-B2 Toll-like receptor 8 (TLR8) specific antagonists and methods of making and uses thereof THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2022-10-11 US disclosed
WO-2012151195-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-11-08 WO disclosed
US-8273742-B2 Disubstituted phthalazine hedgehog pathway antagonists ELI LILLY AND COMPANY (US) 2012-09-25 US disclosed
CN-102459233-A Disubstituted phthalazine hedgehog pathway antagonists LILLY CO ELI (US) 2012-05-16 CN disclosed
EP-2443104-A1 DISUBSTITUTED PHTHALAZINE HEDGEHOG PATHWAY ANTAGONISTS Eli Lilly and Company (US) 2012-04-25 EP disclosed
EP-1505963-B9 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-09-21 EP disclosed
EP-1505963-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-04-20 EP disclosed
US-20100324048-A1 DISUBSTITUTED PHTHALAZINE HEDGEHOG PATHWAY ANTAGONISTS ELI LILLY AND COMPANY (US) 2010-12-23 US disclosed
WO-2010147917-A1 DISUBSTITUTED PHTHALAZINE HEDGEHOG PATHWAY ANTAGONISTS ELI LILLY AND COMPANY (US) 2010-12-23 WO disclosed
WO-2003099274-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324048-A1 DISUBSTITUTED PHTHALAZINE HEDGEHOG PATHWAY ANTAGONISTS SHH, GLI1, SMO GOT1 3692/4885MAPT 3122/4885ALDH1A1 2679/4885
US-20190298717-A1 Hydralazine and Active Derivatives Thereof for Neuronal Cell Survival and Regeneration GSK3B, MAPT, GSK3A GOT1 543/4885MAPT 2/4885ALDH1A1 1374/4885
US-20230132035-A1 Toll-Like Receptor 8 (TLR8)-Specific Antagonists and Methods of Making and Uses Thereof TLR8, TLR3, TLR9 GOT1 2941/4885MAPT 4277/4885ALDH1A1 4565/4885
US-11466010-B2 Toll-like receptor 8 (TLR8) specific antagonists and methods of making and uses thereof TLR8, TLR3, TLR9 GOT1 2762/4885MAPT 4286/4885ALDH1A1 4569/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.