SCHEMBL2126948

SCHEMBL2126948

[CH2].c1ccc(-c2ccc(N3CCN4CCCC(C4)C3)nn2)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 6/20 0.52
HTR3A P46098 1/20 0.52
CHRNB4 P30926 1/20 0.52
CHRNA3 P32297 1/20 0.52
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
RAB9A P51151 1/20 0.45
NFKB2 Q00653 1/20 0.45
KMT2A Q03164 1/20 0.45
RELA Q04206 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3778633 0.86 NPC1 (0.44) CHRNA7HTR3ACHRNB4CHRNA3KDM4E
SCHEMBL2126814 0.79 CYP1A2 (0.50) CHRNB4CHRNA3MEN1ALDH1A1KMT2A
SCHEMBL2124934 0.78 CHRNA7 (0.53) CHRNA7
SCHEMBL5111037 0.77 CHRNA7 (0.51) CHRNA7HTR3ACHRNB4CHRNA3KDM4E
SCHEMBL2124990 0.74 ACHE (0.49) CHRNA7KDM4ENPC1MAPTRAB9A
SCHEMBL5109973 0.74 CHRNA7 (0.50) CHRNA7HTR3ACHRNB4CHRNA3KDM4E
SCHEMBL5832115 0.72 CHRNA7 (0.55) CHRNA7HTR3ACHRNB4CHRNA3KDM4E
SCHEMBL1752797 0.72 CHRNA7 (0.66) CHRNA7HTR3ACHRNB4CHRNA3KDM4E
SCHEMBL6201547 0.72 CHRNA7 (0.74) CHRNA7HTR3ACHRNB4CHRNA3
SCHEMBL5112373 0.72 CHRNA7 (0.48) CHRNA7HTR3ACHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443122-A1 DIAZAHOMOADAMANTANE DERIVATIVES AND METHODS OF USE THEREOF Abbott Laboratories (US) 2012-04-25 EP disclosed
WO-2010145208-A1 DIAZAHOMOADAMANTANE DERIVATIVES AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-12-23 WO disclosed