SCHEMBL2127685

SCHEMBL2127685

CC[C@](C(=O)O)(c1ccccc1)N1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.50
CHRM3 P20309 6/20 0.43
CYP2D6 P10635 3/20 0.41
CHRM2 P08172 3/20 0.41
CHRM1 P11229 3/20 0.41
OPRM1 P35372 3/20 0.41
KCNH2 Q12809 3/20 0.41
HTR1A P08908 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HTR2A P28223 2/20 0.39
DRD3 P35462 2/20 0.39
MLNR O43193 1/20 0.39
HTR2C P28335 1/20 0.39
HRH1 P35367 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CACNA1C Q13936 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2128439 1.00 CYP2B6 (0.50) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL7126061 0.85 CYP2B6 (0.45) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL18112743 0.83 CYP2B6 (0.41) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL327106 0.83 CYP2B6 (0.45) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL703097 0.81 CYP2B6 (0.44) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL4901870 0.79 CYP2B6 (0.45) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL20487815 0.77 CHRM3 (0.41) CHRM3CHRM2CHRM1OPRM1KCNH2
SCHEMBL5816021 0.77 CYP2B6 (0.43) CYP2B6CHRM3CYP2D6CHRM2CHRM1
SCHEMBL7965625 0.75 NPC1 (0.43) CYP2B6CHRM3CYP2D6LMNAMAPK1
SCHEMBL3043721 0.75 CYP2B6 (0.59) CYP2B6CHRM3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121137-B1 QUINUCLIDINOL DERIVATIVES AS MUSCARINIC RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2012-04-25 EP disclosed