SCHEMBL2128199

SCHEMBL2128199

Cc1cccc(N(C)c2cccnc2)n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.47
GRM5 P41594 6/20 0.43
KCNA5 P22460 2/20 0.39
SYK P43405 1/20 0.39
KDM4C Q9H3R0 2/20 0.37
KDM6B O15054 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
CCR1 P32246 1/20 0.35
CCR8 P51685 1/20 0.35
NOTUM Q6P988 1/20 0.35
CYP2E1 P05181 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2131477 0.81 CHRM5 (0.43) CYP2A6GRM5KDM4CKDM6BCCR1
SCHEMBL2130904 0.80 DHFR (0.47) GRM5CCR1CCR8CYP3A4CYP2C9
SCHEMBL10094541 0.80 KCNA5 (0.39) CYP2A6GRM5KCNA5SYKKDM4C
SCHEMBL3409401 0.78 KCNA5 (0.49) CYP2A6GRM5KCNA5CHRNB2CHRNA4
SCHEMBL13443083 0.76 KCNA5 (0.47) CYP2A6GRM5KCNA5SYKKDM4C
Hydrochloric Acid SCHEMBL4024971 0.76 KCNA5 (0.47) CYP2A6GRM5KCNA5CHRNB2CHRNA4
SCHEMBL13957483 0.73 CFTR (0.42) CYP2A6GRM5KCNA5
SCHEMBL12983823 0.73 SYK (0.44) GRM5KCNA5SYKKDM4CKDM6B
SCHEMBL13367476 0.72 KDM4C (0.44) CYP2A6GRM5KCNA5KDM4C
SCHEMBL5075470 0.72 KCNA5 (0.50) CYP2A6GRM5KCNA5CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120101079-A1 SUBSTITUTED 6-AMINO-NICOTINAMIDES AS KCNQ2/3 MODULATORS GRUNENTHAL GMBH (DE) 2012-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101079-A1 SUBSTITUTED 6-AMINO-NICOTINAMIDES AS KCNQ2/3 MODULATORS KCNQ2, KCNQ1, KCNQ3 CYP2A6 440/4885GRM5 1283/4885KCNA5 41/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.