SCHEMBL2128328

SCHEMBL2128328

CC(C)(C)C1[C@@H](Nc2nc(Cl)ncc2F)CCCN1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.46
EGFR P00533 7/20 0.34
BTK Q06187 3/20 0.34
ITK Q08881 2/20 0.34
HCRTR2 O43614 3/20 0.33
HCRTR1 O43613 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2128491 0.79 GSK3A (0.51)
SCHEMBL22496896 0.79 BTK (0.41) BTK
SCHEMBL19665668 0.78 PIN1 (0.42) KMT2AL3MBTL1
SCHEMBL22496836 0.77 JAK3 (0.44) BTK
SCHEMBL22496751 0.77 JAK3 (0.42) EGFRBTK
SCHEMBL17536544 0.77 ALDH1A1 (0.38) HCRTR2HCRTR1ALDH1A1
SCHEMBL22496736 0.76 JAK3 (0.38) BTK
SCHEMBL22496978 0.76 JAK3 (0.32) BTK
SCHEMBL26628895 0.76 MAPK3 (0.40) HCRTR2HCRTR1
SCHEMBL22496852 0.75 JAK3 (0.31) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2442809-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION Vertex Pharmaceuticals Incorporated (US) 2012-04-25 EP disclosed