SCHEMBL2128506

SCHEMBL2128506

COc1c(C(=O)NC2CC2)cc(-c2ccc[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.51
CNR1 P21554 14/20 0.46
CNR2 P34972 14/20 0.46
SMYD3 Q9H7B4 1/20 0.44
CD38 P28907 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542600 0.95 CNR1 (0.52) CYP3A4CNR1CNR2ALDH1A1GAA
SCHEMBL1542756 0.94 CYP3A4 (0.48) CYP3A4CNR1CNR2SMYD3
SCHEMBL1543184 0.94 CYP3A4 (0.46) CYP3A4CNR1CNR2SMYD3CD38
SCHEMBL1542602 0.93 CYP3A4 (0.53) CYP3A4CNR1CNR2SMYD3CD38
SCHEMBL1542583 0.93 CYP3A4 (0.47) CYP3A4CNR1CNR2SMYD3
SCHEMBL2127541 0.89 CYP3A4 (0.47) CYP3A4CNR1CNR2SMYD3
SCHEMBL1542529 0.89 MAPK1 (0.51) CYP3A4CNR1CNR2
SCHEMBL1542533 0.89 CYP3A4 (0.47) CYP3A4CNR1CNR2SMYD3
SCHEMBL1542287 0.87 CYP3A4 (0.44) CYP3A4CNR1CNR2
SCHEMBL1542387 0.84 CYP3A4 (0.47) CYP3A4CNR1CNR2SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8273773-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2012-09-25 US claimed
EP-2307372-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2012-04-25 EP claimed
US-20100021423-A1 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC 2010-01-28 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100021423-A1 Heterocyclic antiviral compounds POLR2A, RRM2B, RRP1B CYP3A4 528/4885CNR1 1007/4885CNR2 1996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.